Pyrazolam powder (CAS Number 39243-02-2)

Pyrazolam powder (CAS Number: 39243-02-2): The Rediscovered Benzodiazepine With Metabolism-Free Effects

So you’ve heard the chatter about Pyrazolam powder (CAS Number: 39243-02-2) and are curious to learn more about this rediscovered benzodiazepine that’s been making waves in recent years. Unlike the benzos you’re probably familiar with, like Xanax or Valium, pyrazolam isn’t metabolized in the body and instead passes through your system unchanged. Developed in the 1970s but largely forgotten, pyrazolam has been experiencing a resurgence as a designer drug that can produce potent sedative and anxiolytic effects. If you’re interested in a benzo experience free from the dulling effects of metabolization, pyrazolam may be worth exploring. But tread carefully, as very little is still known about the long term effects of this mysterious compound. Buy Pyrazolam powder

What Is Pyrazolam powder (CAS 39243-02-2)? A Brief History

Pyrazolam powder (CAS Number: 39243-02-2) is a benzodiazepine that was first developed in the 1970s. Originally created by Leo Sternbach and his team at Hoffman-La Roche, pyrazolam has been rediscovered in recent years and sold as a designer drug.

 

Property Value
Name Pyrazolam
IUPAC name 8-Bromo-1-methyl-6-(pyridin-2-yl)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine
CAS Number 39243-02-2
PubChem CID 12562545
ChemSpider 15417688
Formula C16H12BrN5
Molar mass 354.211 g·mol−1
SMILES CC1=NN=C2CN=C(C3=NC=CC=C3)C3=CC(Br)=CC=C3N12
InChI InChI=1S/C16H12BrN5/c1-10-20-21-15-9-19-16(13-4-2-3-7-18-13)12-8-11(17)5-6-14(12)22(10)15/h2-8H,9H2,1H3
Key BGRWSFIQQPVEML-UHFFFAOYSA-N
Elimination half-life 17 hours
Purity ≥98%

 

Pyrazolam is structurally similar to other benzos like alprazolam (Xanax) and bromazepam (Lexotan). However, unlike most benzodiazepines, pyrazolam seems to not undergo metabolism in the body. Instead, it is excreted unchanged in the urine. This means the effects may last longer and the risk of accumulation could be higher.

Some key points about pyrazolam:

  • It’s a potent anxiolytic, meaning it reduces anxiety and stress.
  • The effects tend to be noticed within 30 minutes of ingestion and last 6-10 hours.
  • The typical dose range is 0.5 mg to 2 mg. Higher doses increase the risks without added benefits.
  • Withdrawal symptoms may occur if used long-term or in high doses. Tapering is recommended.
  • Little is known about the long term effects since it’s an unresearched designer drug. Use with caution.

How Pyrazolam Works: Structural Similarities to Alprazolam and Bromazepam

Pyrazolam works similarly to other benzodiazepines like alprazolam (Xanax) and bromazepam (Lexotan) by binding to benzodiazepine receptors in the brain that regulate gamma-aminobutyric acid (GABA), an inhibitory neurotransmitter. This action promotes relaxation, reduces anxiety and stress, and can induce sedation or sleepiness.

Pyrazolam effects

The primary effects of pyrazolam are:

  • Decreased anxiety and stress
  • Improved mood
  • Sedation and drowsiness
  • Muscle relaxation
  • Amnesia and impaired memory (at high doses)

The effects tend to be less sedating and hypnotic than other benzos like diazepam or clonazepam. The duration of effects is around 6-8 hours.

How Pyrazolam Differs

Unlike most benzodiazepines, pyrazolam does not appear to undergo metabolism in the liver and is instead excreted unchanged in the urine. This means its effects may last longer and remain at a consistent level in the body. Some people report the effects of a single dose of pyrazolam lasting up to 12 hours.

The lack of metabolism also means pyrazolam may have a lower potential for interaction with other drugs and supplements compared to benzodiazepines which are broken down in the liver. However, more research is still needed to confirm this.

In studies, pyrazolam demonstrated anxiolytic, anticonvulsant, muscle relaxant, and sedative effects. It may help relieve symptoms of anxiety disorders, insomnia, seizures, and muscle spasms. The potency of pyrazolam seems to be similar to or slightly higher than diazepam (Valium) and alprazolam.

While pyrazolam shows promise as an alternative to traditional benzodiazepines, its legal status remains unclear in many places. Some countries have banned pyrazolam, classifying it as an illegal narcotic. If considering pyrazolam, check your local laws and consult a doctor.

Why Pyrazolam Is Unique: Lack of Metabolism

Pyrazolam is unique among benzodiazepines in that it is not metabolized in the body. Most benzodiazepines are broken down into other compounds by enzymes in the liver, which can alter their effects and duration of action. Pyrazolam, on the other hand, is excreted from the body unchanged in urine.

This lack of metabolism is thought to explain why the effects of pyrazolam seem to be relatively consistent and long-lasting compared to other benzos. The typical elimination half-life of pyrazolam is over 12 hours, meaning it can continue to produce effects for up to a day after dosing. The duration of noticeable effects seems to be 6-12 hours for most people.

Some key points about pyrazolam’s metabolism-free nature:

  1. The potency and effects are not altered by individual differences in liver enzyme function. The effects tend to be the same from person to person.
  2. There are no active metabolites produced that could have unintended effects or interact with other drugs. What you ingest is what you get.
  3. The lack of metabolism may allow for simpler dosing and less risk of overdose due to drug interactions.
  4. The long duration of effects could increase risks associated with redosing or combining with other CNS depressants. Caution is advised.

While pyrazolam’s lack of metabolism makes it unique, it does not necessarily make it safer than other benzodiazepines. Responsible and informed use is still critical to avoiding potentially serious risks.

Where to Buy Pyrazolam in USA: Finding a Reputable Vendor

So you’re interested in pyrazolam, a rediscovered benzodiazepine with some unique properties. Before you buy pyrazolam powder or pills online, it’s important to find a reputable vendor.

FAQ

What is pyrazolam and how does it work?

Pyrazolam is a benzodiazepine, similar in structure to Xanax (alprazolam) and Lexotan (bromazepam). Like other benzos, it works by binding to GABA receptors in the brain, slowing activity in the central nervous system. This produces effects like anxiety relief, sedation, and muscle relaxation.

Is pyrazolam legal?

Pyrazolam is currently unregulated in many parts of the world, though some countries have banned it. In the US, pyrazolam is not approved for medical use and is considered an unscheduled research chemical. Possession or sale for human consumption may be prosecuted under the Federal Analog Act. Check your local laws before purchasing.

What’s the typical dosage for pyrazolam?

Pyrazolam comes in powder or pellet form. An average dose for anxiety relief and sedation is 0.5-2 mg. Start with 0.5 mg and wait at least 2 hours before increasing the dose. Doses over 2 mg greatly increase the risks of side effects like amnesia, impaired motor function, and overdose.

Is pyrazolam addictive?

Yes, like other benzodiazepines, pyrazolam can be addictive if misused. It should only be taken occasionally and at the lowest effective dose. Do not take pyrazolam daily or in high doses, as this can lead to physical dependence and difficult withdrawal.

Read more :

Highly potent designer benzodiazepines

Rilmazafone Half-Life Explained: What You Need to Know

Risk of Dependence and Addiction to Benzodiazepines

The Benefits of Research Chemicals: Your Guide to Learning More

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